Peficitinib (ASP-015K)

Name: Peficitinib (ASP-015K); MyBioSource
Brand: MyBioSource
SKU: MBS3606755
Price: 220 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3606755

Peficitinib (ASP-015K, JNJ-54781532) is a potent JAK inhibitor with IC50s of 3.9 and 0.7 nM for JAK1 and JAK3 respectively; inhibits IL-2-dependent T cell proliferation in vitro and STAT5 phosphorylation in vitro and ex vivo. More details

$220 / 2 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Peficitinib, Biochemical

Full Product Name

Peficitinib

Product Synonym Names

ASP-015K; JNJ-54781532

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

326.3929

Suitability

DMSO: >=60mg/mL

Target

JAK

Receptor

JAK

Chemical Name

1H-Pyrrolo[2, 3-b]pyridine-5-carboxamide, 4-[(5-hydroxytricyclo[3.3.1.13, 7]dec-2-yl)amino]-, stereoisomer

SMILES

C1C2CC3CC(C2)(CC1C3NC4=C5C=CNC5=NC=C4C(=O)N)O

Molecular Formula

C18H22N4O2

CAS Number

944118-01-8

Product Categories/Family for Peficitinib biochemical

Rheumatoid Arthritis; Angiogenesis; Inflammation/Immunology

Product References and Citations for Peficitinib biochemical

1. Oda K, et al. Xenobiotica. 2015; 45 (6):488-94.
2. Takeuchi T, et al. Ann Rheum Dis. 2016 Jun; 75 (6):1057-64.

Other Notes

Small volumes of Peficitinib biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Peficitinib purchase

MBS3606755 is a biochemical targeting Peficitinib.