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KDM5A covalent inhibitor N71

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3607066

KDM5A covalent inhibitor N71 is an irreversible KDM5A inhibitor (IC50=0.22 uM) that covalently interacts with Cys481. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
KDM5A covalent inhibitor N71, Biochemical
Full Product Name
KDM5A covalent inhibitor N71
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
522.664
Target
Histone Demethylase
Receptor
Histone Demethylase
Chemical Name
(E)-2-((3-(4-(dimethylamino)but-2-enamido)phenyl)(2-(piperidin-1-yl)ethoxy)methyl)thieno[3, 2-b]pyridine-7-carboxylic acid
Molecular Formula
C28H34N4O4S

Product Categories/Family for KDM5A covalent inhibitor N71 biochemical

Chromatin/Epigenetic

Structure of KDM5A covalent inhibitor N71 biochemical

KDM5A covalent inhibitor N71 Biochemical – Cat# MBS3607066

Product References and Citations for KDM5A covalent inhibitor N71 biochemical

1. Horton JR, et al. J Med Chem. 2018 Nov 15. doi: 10.1021/acs.jmedchem.8b01219.

Other Notes

Small volumes of KDM5A covalent inhibitor N71 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for KDM5A covalent inhibitor N71 purchase

MBS3607066 is a biochemical targeting KDM5A covalent inhibitor N71.
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