Uprosertib

Name: Uprosertib; MyBioSource
Brand: MyBioSource
SKU: MBS3607117
Price: 240 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3607117

Uprosertib (GSK2141795) is a selective, ATP-competitive, and orally bioavailable Akt inhibitor with IC50 of 180 nM, 328 nM, and 38 nM for Akt 1, 2 and 3, respectively. Phase 2. More details

$240 / 2 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Uprosertib, Biochemical

Full Product Name

Uprosertib

Product Synonym Names

GSK2141795, GSK 795, Uprosertib

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

429.25

Suitability

DMSO: >=150mg/mL (349.45mM)
H2O: <0.1mg/mL

Target

Transaminase

Receptor

Akt1; Akt2; Akt3

Chemical Name

N-((S)-1-amino-3-(3, 4-difluorophenyl)propan-2-yl)-5-chloro-4-(4-chloro-1-methyl-1H-pyrazol-5-yl)furan-2-carboxamide

SMILES

Cn1c(c(cn1)Cl)c1c(oc(c1)C(=O)N[C@@H](Cc1cc(c(cc1)F)F)CN)Cl

Molecular Formula

C18H16Cl2F2N4O2

CAS Number

1047634-65-0

Product Categories/Family for Uprosertib biochemical

Cancer

Product References and Citations for Uprosertib biochemical

1.Pachl F, et al. Characterization of a chemical affinity probe targeting Akt kinases. J Proteome Res. 2013 Aug 2; 12 (8):3792-800.

Other Notes

Small volumes of Uprosertib biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Uprosertib purchase

MBS3607117 is a biochemical targeting Uprosertib.

Uprosertib

Product Overview

Product Categories/Family for Uprosertib biochemical

Structure of Uprosertib biochemical

Related Product Information for Uprosertib biochemical

Product References and Citations for Uprosertib biochemical

Other Notes

Searchable Terms for Uprosertib purchase