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G007-LK

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3607264

G007-LK is a selective inhibitor of TNKS1 and TNKS2, with IC50s of 46 nM and 25 nM, respectively. More details

$250 / 2 mg +1 FREE 8GB USB
Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
G007-LK, Biochemical
Full Product Name
G007-LK
Product Synonym Names
G007LK; G007LK; G007 LK
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
529.96
Suitability
DMSO: >=30mg/mL (56.61mM)
Target
AChR
Receptor
TNKS1; TNKS2
Chemical Name
(E)-4-(5-(2-(4-(2-chlorophenyl)-5-(5-(methylsulfonyl)pyridin-2-yl)-4H-1, 2, 4-triazol-3-yl)vinyl)-1, 3, 4-oxadiazol-2-yl)benzonitrile
SMILES
CS(=O)(=O)c1cnc(cc1)c1nnc(n1c1ccccc1Cl)/C=C/c1nnc(o1)c1ccc(cc1)C#N
Molecular Formula
C25H16ClN7O3S
CAS Number
1380672-07-0

Product Categories/Family for G007-LK biochemical

Endocrinology/Hormones; Cancer

Structure of G007-LK biochemical

G007-LK Biochemical – Cat# MBS3607264

Product References and Citations for G007-LK biochemical

1.Voronkov A, etal.Structural basis and SAR for G007-LK, a lead stage 1, 2, 4-triazole based specific tankyrase 1/2 inhibitor.J Med Chem. 2013 Apr 11; 56 (7):3012-23.

Other Notes

Small volumes of G007-LK biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for G007-LK purchase

MBS3607264 is a biochemical targeting G007-LK.
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