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CPI-169

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3607299

CPI-169 is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and 6.1 nM for EZH2 WT, EZH2 Y641N, and EZH1, respectively. More details

$255 / 2 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
CPI-169, Biochemical
Full Product Name
CPI-169
Product Synonym Names
CPI-169; CPI 169; CPI169
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
528.66
Suitability
DMSO: >=59mg/mL (111.60mM)
Target
ALK
Receptor
EZH1; EZH2 WT; EZH2 Y641N
Chemical Name
(R, Z)-1-(1-(1-(ethylsulfonyl)piperidin-4-yl)ethyl)-N-((2-hydroxy-4-methoxy-6-methylpyridin-3-yl)methyl)-2-methyl-1H-indole-3-carbimidic acid
SMILES
CCS(=O)(=O)N1CCC(CC1)C(C)n1c2ccccc2c(C(=O)NCc2c(OC)cc(C)[nH]c2=O)c1C
Molecular Formula
C27H36N4O5S
CAS Number
1450655-76-1

Product Categories/Family for CPI-169 biochemical

Structure of CPI-169 biochemical

CPI-169 Biochemical – Cat# MBS3607299

Product References and Citations for CPI-169 biochemical

1.Bradley WD, etal.EZH2 inhibitor efficacy in non-Hodgkin's lymphoma does not require suppression of H3K27 monomethylation.Chem Biol. 2014 Nov 20; 21 (11):1463-75.

Other Notes

Small volumes of CPI-169 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for CPI-169 purchase

MBS3607299 is a biochemical targeting CPI-169.
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