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Entospletinib

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3607889

Entospletinib ?IC50= 7.7 nM?is a specific Syk inhibitor, which is orally bioavailable. More details

$235 / 2 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Entospletinib, Biochemical
Full Product Name
Entospletinib
Product Synonym Names
Entospletinib; GS9973; GS 9973
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
411.47
Suitability
DMSO: >=43mg/mL (104.51mM)
Target
Antibacterial
Receptor
Syk
Chemical Name
6-(1H-indazol-6-yl)-N-(4-morpholinophenyl)imidazo[1, 2-a]pyrazin-8-amine
SMILES
C1CN(CCO1)c1ccc(Nc2nc(cn3ccnc23)c2ccc3cn[nH]c3c2)cc1
Molecular Formula
C23H21N7O
CAS Number
1229208-44-9

Product Categories/Family for Entospletinib biochemical

GPCR/G Protein; Cancer

Structure of Entospletinib biochemical

Entospletinib Biochemical – Cat# MBS3607889

Product References and Citations for Entospletinib biochemical

1.Currie KS, et al. Discovery of GS-9973, a Selective and Orally Efficacious Inhibitor of Spleen Tyrosine Kinase. J Med Chem. 2014 May 8; 57 (9):3856-73.

Other Notes

Small volumes of Entospletinib biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Entospletinib purchase

MBS3607889 is a biochemical targeting Entospletinib.
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