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Theliatinib

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3610697

Theliatinib a potent and highly selective EGFR inhibitor with anti-tumor activity. Ki of 0.05 nM for wild type EGFR and IC50s of 3 and 22 nM for EGFR and EGFR T790M/L858R mutant respectively. More details

$300 / 5 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Theliatinib, Biochemical
Full Product Name
Theliatinib
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
442.5
Suitability
DMSO: 47mg/mL (106.21mM)
Target
EGFR
Receptor
EGFR
Chemical Name
(3aR6aR)-N-(4-((3-ethynylphenyl)amino)-7-methoxyquinazolin-6-yl)-1-methylhexahydropyrrolo[34-b]pyrrole-5(1H)-carboxamide
SMILES
[H][C@]12CCN(C)[C@@]1([H])CN(C2)C(=O)Nc1cc2c(Nc3cccc(c3)C#C)ncnc2cc1OC
Molecular Formula
C25H26N6O2
CAS Number
1353644-70-8

Product Categories/Family for Theliatinib biochemical

Angiogenesis

Structure of Theliatinib biochemical

Theliatinib Biochemical – Cat# MBS3610697

Product References and Citations for Theliatinib biochemical

1.Ren Y Zheng J Fan S et al. Anti-tumor efficacy of theliatinib in esophageal cancer patient-derived xenografts models with epidermal growth factor receptor (EGFR) overexpression and gene amplification. [J]. Oncotarget 2017 8 (31):50832-50844.

Other Notes

Small volumes of Theliatinib biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Theliatinib purchase

MBS3610697 is a biochemical targeting Theliatinib.
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