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BQR-695 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5750082

MBS5750082 is an inhibitor targeting BQR-695. Also known as BQR-695 (Synonyms: NVP-BQR695). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
BQR-695, Inhibitor
Full Product Name
BQR-695 (Synonyms: NVP-BQR695)
Product Gene Name
BQR-695, inhibitor
Product Synonym Names
NVP-BQR695
Form/Format
POWDER
Purity/Purification
99.0%
Preparation and Storage
For 3 years at -20 degree C (powder)
For 2 years -80 degree C in solvent.
Molecular Weight
352.394
CAS
1513879-21-4
Formula
C19H20N4O3
Pathways
PI3K/Akt/mTOR signaling
Target
Plasmodium PI4KIIIbeta; human PI4KIIIbeta
Smiles
CNC(=O)CNc1cnc2ccc(cc2n1)c1cc(c(cc1)OC)OC
Receptor
PI3KIIIbeta
Bioactivity
BQR-695 is a phosphatidylinositol 4-kinase (PI4K) inhibitor with IC50s of 80 and 3.5 nM for human PI4KIIIbeta and Plasmodium variant of PI4KIIIbeta, respectively.
Solubility Note
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Product References and Citations for BQR-695, inhibitor

1. Fowler ML, et al. Using hydrogen deuterium exchange mass spectrometry to engineer optimized constructs for crystallization of protein complexes: Case study of PI4KIIIbeta with Rab11. Protein Sci. 2016 Apr; 25 (4):826-39.

Other Notes

Small volumes of BQR-695, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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