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ASP-9521 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5750119

MBS5750119 is an inhibitor targeting ASP-9521. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
ASP-9521, Inhibitor
Full Product Name
ASP-9521
Product Gene Name
ASP-9521, inhibitor
Form/Format
POWDER
Purity/Purification
95.1%
Preparation and Storage
For 3 years at -20 degree C (powder)
For 2 years -80 degree C in solvent.
Molecular Weight
330.32
CAS
1126084-37-4
Formula
C19H26N2O3
Pathways
Metabolism
Target
AKR1C3
Smiles
CC(C)(CC1CCN(CC1)C(=O)c1cc2c([nH]1)ccc(c2)OC)O
Receptor
AKR1C3
Bioactivity
ASP-9521 is a potent, selective and orally available AKR1C3 inhibitor with an IC50 of 11 nM for human AKR1C3.
Solubility Note
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Structure of ASP-9521, inhibitor

ASP-9521 Inhibitor – Cat# MBS5750119

Product References and Citations for ASP-9521, inhibitor

1. Kikuchi A, et al. In vitro and in vivo characterisation of ASP9521: a novel, selective, orally bioavailable inhibitor of 17beta-hydroxysteroid dehydrogenase type 5 (17betaHSD5; AKR1C3).Invest New Drugs. 2014 Oct; 32 (5):860-70.

Other Notes

Small volumes of ASP-9521, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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