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EPZ020411 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5750455

MBS5750455 is an inhibitor targeting EPZ020411. EPZ020411 is a specific and effective inhibitor of PRMT6 (IC50=10 nM). More details

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Product Documentation
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Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
EPZ020411, Inhibitor
Full Product Name
EPZ020411
Product Gene Name
EPZ020411, inhibitor
Product Synonym Names
Histone Methyltransferase
Form/Format
POWDER
Purity/Purification
98.00%
Preparation and Storage
Powder: 3 years -20 degree C
In Solvent: 2 years -80 degree C
Molecular Weight
442.6
CAS Number
1700663-41-7
Formula
C25H38N4O3
Smiles
CNCCN(C)Cc1c[nH]nc1-c1ccc(O[C@H]2C[C@@H](C2)OCCC2CCOCC2)cc1
Solubility
DMSO: 10 mM
Pathways
Chromatin; Epigenetic
Receptor
PRMT6
Product Remark
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Product Categories/Family for EPZ020411, inhibitor

Cancer

Chemical Structure of EPZ020411, inhibitor

EPZ020411 Inhibitor – Cat# MBS5750455

Product References and Citations for EPZ020411, inhibitor

1. Mitchell LH, et al. Aryl Pyrazoles as Potent Inhibitors of Arginine Methyltransferases: Identification of the First PRMT6 ToolCompound. ACS Med Chem Lett. 2015 Apr 6; 6(6):655-659.

Other Notes

Small volumes of EPZ020411, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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