GSK2879552 2HCl Inhibitor

Name: GSK2879552 2HCl Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5750537
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5750537

GSK2879552 is an orally available, irreversible inhibitor of lysine specific demethylase 1 (LSD1), with potential antineoplastic activity. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

GSK2879552 2HCl, Inhibitor

Full Product Name

GSK2879552 2HCl (1401966-69-5(Free Base))

Product Synonym Names

Histone Demethylase

Form/Format

POWDER

Purity/Purification

99.9%

Preparation and Storage

Powder: 3 years -20 degree C
In Solvent: 2 years -80 degree C

Molecular Weight

437.41

CAS Number

1401966-69-5 (Free Base)

Formula

C23H30Cl2N2O2

Smiles

Cl.Cl.OC(=O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1

Solubility

DMSO: 4.37 mg/mL (10 mM)

Pathways

Chromatin; Epigenetic

Receptor

LSD1

Product Remark

For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Product Categories/Family for GSK2879552 2HCl, inhibitor

Cancer

Product References and Citations for GSK2879552 2HCl, inhibitor

1. Huang M,etal.Targeting KDM1A attenuates Wnt/beta-catenin signaling pathway to eliminate sorafenib-resistant stem-like cells in hepatocellular carcinoma.Cancer Lett. 2017 Jul 10; 398:12-21.

Other Notes

Small volumes of GSK2879552 2HCl, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GSK2879552 2HCl purchase

MBS5750537 is an inhibitor targeting GSK2879552 2HCl. Also known as GSK2879552 2HCl (1401966-69-5(Free Base)).