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Saclofen Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5750554

Saclofen is a sulfonic analog of the inhibitory neurotransmitter gamma-aminobutyric acid (GABA) that acts as a competitive antagonist of the GABAB receptor (IC50: 7.8 uM).1 This compound can be used to determine the functional roles for the GABAB receptor as… More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Product Overview

Online Datasheet in PDF
Product Name
Saclofen, Inhibitor
Full Product Name
Saclofen
Product Synonym Names
GABA Receptor
Form/Format
POWDER
Purity/Purification
98.0%
Preparation and Storage
Powder: 3 years -20 degree C
In Solvent: 2 years -80 degree C
Molecular Weight
249.71
CAS Number
125464-42-8
Formula
C9H12ClNO3S
Smiles
NCC(CS(O)(=O)=O)c1ccc(Cl)cc1
Solubility
DMSO: 0.3 mg/mL; Water: 10 mM
Pathways
Membrane Transporter; Ion Channel
Receptor
GABAB
Product Remark
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Chemical Structure of Saclofen, inhibitor

Saclofen Inhibitor – Cat# MBS5750554

Product References and Citations for Saclofen, inhibitor

1. Drew C A, Johnston G A R, Kerr D I B, et al. Inhibition of baclofen binding to rat cerebellar membranes by phaclofen, saclofen, 3-aminopropylphosphonic acid and related GABAB receptor antagonists[J]. Neuroscience letters, 1990, 113(1): 107-110.

Other Notes

Small volumes of Saclofen, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Saclofen purchase

MBS5750554 is an inhibitor targeting Saclofen.
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