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PF-01247324 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5750592

PF-01247324 is a selective and orally bioavailable Nav1.8 channel blocker (IC50: 196 nM). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
PF-01247324, Inhibitor
Full Product Name
PF-01247324
Product Gene Name
PF-01247324, inhibitor
Product Synonym Names
Sodium Channel blocker
Form/Format
POWDER
Purity/Purification
98.00%
Preparation and Storage
Powder: 3 years -20 degree C
In Solvent: 2 years -80 degree C
Molecular Weight
330.6
CAS Number
875051-72-2
Formula
C13H10Cl3N3O
Smiles
CNC(=O)c1ccc(c(N)n1)-c1cc(Cl)cc(Cl)c1Cl
Solubility
DMSO: 30 mg/mL
Pathways
Membrane Transporter; Ion Channel
Receptor
Na(V1.8) channel
Product Remark
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Chemical Structure of PF-01247324, inhibitor

PF-01247324 Inhibitor – Cat# MBS5750592

Product References and Citations for PF-01247324, inhibitor

1. Payne CE, et al. A novel selective and orally bioavailable Nav 1.8 channel blocker, PF-01247324, attenuates nociception and sensory neuron excitability. Br J Pharmacol. 2015 May; 172(10):2654-70.

Other Notes

Small volumes of PF-01247324, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for PF-01247324 purchase

MBS5750592 is an inhibitor targeting PF-01247324.
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