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TCS-OX2-29 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5750769

TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
TCS-OX2-29, Inhibitor
Full Product Name
TCS-OX2-29
Product Gene Name
TCS-OX2-29, inhibitor
Product Synonym Names
OX Receptor
Form/Format
POWDER
Purity/Purification
98.00%
Preparation and Storage
Powder: 3 years -20 degree C
In Solvent: 2 years -80 degree C
Molecular Weight
397.51
CAS Number
372523-75-6
Formula
C23H31N3O3
Smiles
COc1cc2CCN(Cc2cc1OC)C(=O)[C@@H](NCc1ccncc1)C(C)(C)C
Solubility
DMSO: 10 mM
Pathways
GPCR; G Protein
Receptor
OX2
Product Remark
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Chemical Structure of TCS-OX2-29, inhibitor

TCS-OX2-29 Inhibitor – Cat# MBS5750769

Product References and Citations for TCS-OX2-29, inhibitor

1. Hirose M et al. N-acyl 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline: the first orexin-2 receptor selective non-peptidicantagonist. Bioorg Med Chem Lett, 2003 Dec 15, 13(24):4497-9.

Other Notes

Small volumes of TCS-OX2-29, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for TCS-OX2-29 purchase

MBS5750769 is an inhibitor targeting TCS-OX2-29.
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