Batefenterol Inhibitor

Name: Batefenterol Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5751081
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5751081

Batefenterol (GSK961081, TD-5959) is a muscarinic receptor antagonist and beta2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic and hbeta2-adrenoceptor (Ki:1.4/1.3/3.7 nM). More details

Please Inquire

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Batefenterol, Inhibitor

Full Product Name

Batefenterol

Product Synonym Names

Adrenergic Receptor agonist

Form/Format

POWDER

Purity/Purification

98.00%

Preparation and Storage

Powder: 3 years -20 degree C
In Solvent: 2 years -80 degree C

Molecular Weight

740.24

CAS Number

743461-65-6

Formula

C40H42ClN5O7

Smiles

ClC1=C(N([H])C(CCN2CCC(OC(N(C3=C(C4=CC=CC=C4)C=CC=C3)[H])=O)CC2)=O)C=C(OC)C(CN(C[C@H](O)C5=C(C=CC(N6[H])=O)C6=C(O)C=C5)[H])=C1

Solubility

DMSO: 5 mg/mL; Water: Insoluble

Pathways

GPCR; G Protein

Receptor

beta2-adrenoceptor

Product Remark

For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Product Categories/Family for Batefenterol, inhibitor

Respiratory Disease

Product References and Citations for Batefenterol, inhibitor

1. Hegde SS, et al. Pharmacologic characterization of GSK-961081 (TD-5959), a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and beta2-adrenoceptor agonist properties. J Pharmacol Exp Ther. 2014 Oct; 351(1):190-9.

Other Notes

Small volumes of Batefenterol, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Batefenterol purchase

MBS5751081 is an inhibitor targeting Batefenterol.