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SGC2085 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5751091

SGC2085 is an effective and selective coactivator-associated arginine methyltransferase 1 (CARM1) inhibitor (IC50: 50 nM). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
SGC2085, Inhibitor
Full Product Name
SGC2085
Product Gene Name
SGC2085, inhibitor
Product Synonym Names
Histone Methyltransferase inhibitor
Form/Format
POWDER
Purity/Purification
98.00%
Preparation and Storage
Powder: 3 years -20 degree C
In Solvent: 2 years -80 degree C
Molecular Weight
312.41
CAS Number
1821908-48-8
Formula
C19H24N2O2
Smiles
C[C@H](N)C(=O)NCc2ccc(Oc1cc(C)cc(C)c1)c(C)c2
Solubility
DMSO: 50 mg/mL; Ethanol: 40 mg/mL; Water: Insoluble
Pathways
Chromatin; Epigenetic
Receptor
Coactivator Associated Arginine Methyltransferase 1 (CARM1)
Product Remark
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Product References and Citations for SGC2085, inhibitor

1. Ferreira de Freitas R, et al. Discovery of a Potent and Selective Coactivator Associated Arginine Methyltransferase 1 (CARM1) Inhibitor by Virtual Screening. J Med Chem. 2016 Jul 28; 59(14):6838-47.

Other Notes

Small volumes of SGC2085, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for SGC2085 purchase

MBS5751091 is an inhibitor targeting SGC2085.
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