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TGR-1202 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5751442

MBS5751442 is an inhibitor targeting TGR-1202. TGR-1202 is a PI3Kdelta inhibitor. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
TGR-1202, Inhibitor
Full Product Name
TGR-1202
Product Gene Name
TGR-1202, inhibitor
Product Synonym Names
TGR1202; TGR 1202; RP5264,uMbralisib
Form/Format
Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.
Molecular Weight
571.55
Formula
C31H24F3N5O3
CAS
1532533-67-7
Smiles
CC(C)Oc1ccc(cc1F)-c1nn([C@@H](C)c2oc3ccc(F)cc3c(=O)c2-c2cccc(F)c2)c2ncnc(N)c12
Receptor (IC50)
PI3Kdelta
Solubility
DMSO: 91mg/mL (159.2mM)
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for TGR-1202, inhibitor

Home; PI3K/Akt/mTOR signaling; PI3K

Structure of TGR-1202, inhibitor

TGR-1202 Inhibitor – Cat# MBS5751442

Product References and Citations for TGR-1202, inhibitor

1. Swaroop Vakkalankaa, et al. Inhibition of PI3Kdelta kinase by a selective, small molecule inhibitor suppresses B-cell proliferation and leukemic cell growth.
2. Deng C, et al. Silencing c-Myc translation as a therapeutic strategy through targeting PI3Kdelta and CK1epsilon in hematological malignancies. Blood. 2017 Jan 5;129 (1):88-99

Other Notes

Small volumes of TGR-1202, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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