Leuprolide Acetate Inhibitor

Name: Leuprolide Acetate Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5751494
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5751494

Leuprolide is an agonist at pituitary GnRH receptors. Leuprorelin is a gonadotropin-releasing hormone (GnRH) analog used to treat a wide range of sex hormone-related disorders including advanced prostatic cancer, endometriosis, and precocious puberty.… More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Product Name

Leuprolide Acetate, Inhibitor

Full Product Name

Leuprolide Acetate

Product Synonym Names

Leuprorelin acetate

Form/Format

Powder

Purity/Purification

100.00%

Preparation and Storage

Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Molecular Weight

1269.45

Formula

C59H84N16O12.C2H4O2

CAS

74381-53-6

Smiles

CC(O)=O.CCNC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H]1CCC(=O)N1

Receptor (IC50)

GNRHR

Solubility

DMSO: 40mg/mL
Water: 60mg/mL
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for Leuprolide Acetate, inhibitor

Home; GPCR/G Protein; GNRH Receptor

Product References and Citations for Leuprolide Acetate, inhibitor

1. Wilson AC, et al. Leuprolide acetate: a drug of diverse clinical applications. Expert Opin Investig Drugs. 2007 Nov;16 (11):1851-63.
2. Lama G, et al. Leuprorelin acetate long-lasting effects on GnRH receptors of prostate cancer cells: an atomic force microscopy study of agonist/receptor interaction. PLoS One. 2013;8 (1):e52530.

Other Notes

Small volumes of Leuprolide Acetate, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Leuprolide Acetate purchase

MBS5751494 is an inhibitor targeting Leuprolide Acetate.