BAY-8002 Inhibitor

Name: BAY-8002 Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5751647
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5751647

BAY-8002 is a potent dual MCT1/2 inhibitor (IC50 values are 3, 8, and 12nM at rat (C6), human (DLD-1) and mouse (4T1) MCT1 respectively). More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

BAY-8002, Inhibitor

Full Product Name

BAY-8002

Product Gene Name

BAY-8002, inhibitor

Product Synonym Names

BAY8002; BAY 8002

Form/Format

Powder

Purity/Purification

99.13%

Preparation and Storage

Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Molecular Weight

415.85

Formula

C20H14ClNO5S

CAS

724440-27-1

Smiles

OC(=O)c1ccccc1NC(=O)c1cc(ccc1Cl)S(=O)(=O)c1ccccc1

Receptor (IC50)

MCT1: 85nM (MCT1-expressing DLD-1 cells)

Solubility

DMSO: 50mg/mL, 120.24mM
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for BAY-8002, inhibitor

Home; Membrane transporter/Ion Channel

Product References and Citations for BAY-8002, inhibitor

1. Quanz M, et al. Preclinical Efficacy of the Novel Monocarboxylate Transporter 1 Inhibitor BAY-8002 and Associated Markers of Resistance. Mol Cancer Ther. 2018 Nov;17 (11):2285-2296.

Other Notes

Small volumes of BAY-8002, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for BAY-8002 purchase

MBS5751647 is an inhibitor targeting BAY-8002.