Eprotirome Inhibitor

Name: Eprotirome Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5751782
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5751782

Eprotirome, a synthetic thyroid hormone mimetic, is a thyroid hormone receptor agonist. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Eprotirome, Inhibitor

Full Product Name

Eprotirome

Form/Format

Powder

Purity/Purification

98.25%

Preparation and Storage

Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Molecular Weight

487.14

Formula

C18H17Br2NO5

CAS

355129-15-6

Smiles

CC(C)c1cc(Oc2c(Br)cc(NC(=O)CC(O)=O)cc2Br)ccc1O

Receptor (IC50)

THR

Solubility

DMSO: 90mg/mL, 184.75mM
Ethanol: 30mg/mL
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for Eprotirome, inhibitor

Home; Endocrinology/Hormones; Thyroid hormone receptor (THR)

Product References and Citations for Eprotirome, inhibitor

1. Berkenstam A, et al. The thyroid hormone mimetic compound KB2115 lowers plasma LDL cholesterol and stimulates bile acid synthesis without cardiac effects in humans. Proc Natl Acad Sci U S A. 2008 Jan 15;105 (2):663-7.
2. Martagón AJ, et al. The amelioration of hepatic steatosis by thyroid hormone receptor agonists is insufficient to restore insulin sensitivity in ob/ob mice. PLoS One. 2015 Apr 7;10 (4):e201221987.

Other Notes

Small volumes of Eprotirome, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Eprotirome purchase

MBS5751782 is an inhibitor targeting Eprotirome.