Asapiprant Inhibitor

Name: Asapiprant Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5751799
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5751799

Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44nM). It exhibited high affinity and selectivity for the DP1 receptor. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Asapiprant, Inhibitor

Full Product Name

Asapiprant

Form/Format

Powder

Purity/Purification

99.23%

Preparation and Storage

Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Molecular Weight

501.55

Formula

C24H27N3O7S

CAS

932372-01-5

Smiles

CC(C)Oc1ccc(cc1)S(=O)(=O)N1CCN(CC1)c1ccc(-c2ncco2)c(OCC(O)=O)c1

Receptor (IC50)

DP1 receptor: 0.44nM (Ki)

Solubility

DMSO: 10mg/mL, 19.94mM
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for Asapiprant, inhibitor

Home; GPCR/G Protein; Prostaglandin Receptor

Product References and Citations for Asapiprant, inhibitor

1. Takahashi G, et al. Effect of the potent and selective DP1 receptor antagonist, asapiprant (S-555739), in animal models of allergic rhinitis and allergic asthma. Eur J Pharmacol. 2015 Oct 15;765:15-23.

Other Notes

Small volumes of Asapiprant, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Asapiprant purchase

MBS5751799 is an inhibitor targeting Asapiprant.