CK1-IN-1 Inhibitor

Name: CK1-IN-1 Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5751804
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5751804

CK1-IN-1, compound 1c reported in patent WO2015119579A1, is a casein kinase 1 (CK1) inhibitor. It has IC50s of 15nM, 16nM, 73nM for CK1delta, and CK1epsilon, p38sigma MAPK, respectively. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

CK1-IN-1, Inhibitor

Full Product Name

CK1-IN-1

Product Gene Name

CK1-IN-1, inhibitor

Product Synonym Names

PUN51207

Form/Format

Powder

Purity/Purification

98.79%

Preparation and Storage

Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Molecular Weight

383.39

Formula

C24H15F2N3

CAS

1784751-20-7

Smiles

Fc1ccc(cc1)-c1nc([nH]c1-c1ccncc1)-c1ccc2ccccc2c1F

Receptor (IC50)

CK1delta: 15nM (cell free)
CK1epsilon: 16nM (cell free)
p38sigma MAPK: 73nM (cell free)

Solubility

DMSO: 60mg/mL (156.5mM)
Water: Insoluble
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for CK1-IN-1, inhibitor

Home; Metabolism; Casein Kinase; CK1-IN-1

Product References and Citations for CK1-IN-1, inhibitor

1. Filip LACO,et al. 2,4,5-tri-substituted azole-based casein kinase 1 inhibitors as inducers for cardiomyogenesis. WO2015119579A1.

Other Notes

Small volumes of CK1-IN-1, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for CK1-IN-1 purchase

MBS5751804 is an inhibitor targeting CK1-IN-1.