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PKC-theta Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752164

MBS5752164 is an inhibitor targeting PKC-theta. Also known as PKC-theta inhibitor. PKC-theta inhibitor is a selective PKC-thetainhibitor (IC50:12nM). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
PKC-theta, Inhibitor
Full Product Name
PKC-theta inhibitor
Form/Format
Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.
Molecular Weight
454.4
Formula
C20H25F3N6O3
CAS
736048-65-0
Smiles
Cl.NCC1CCC(CNc2nc(NCc3ccccc3OC(F)(F)F)ncc2[N+]([O-])=O)CC1
Receptor (IC50)
PKC-theta: 12nM
Solubility
DMSO: 62.5mg/mL (137.53mM)
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for PKC-theta, inhibitor

Home; Cytoskeletal Signaling; PKC; PKC-theta inhibitor

Structure of PKC-theta, inhibitor

PKC-theta Inhibitor – Cat# MBS5752164

Product References and Citations for PKC-theta, inhibitor

1. Cywin C L, Dahmann G, Iii A S P, et al. Discovery of potent and selective PKC-theta inhibitors[J]. Bioorganic & Medicinal Chemistry Letters, 2007, 17 (1):225-230.

Other Notes

Small volumes of PKC-theta, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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