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PI3Kdelta1 Inhibitor – Pi3kdelta 1

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752176

MBS5752176 is an inhibitor targeting PI3Kdelta1. Also known as Selective PI3Kdelta Inhibitor 1. Selective PI3Kdelta Inhibitor 1 is a PI3Kdelta Inhibitor (IC50 = 0.9nM). More details

Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
PI3Kdelta 1 (PI3Kdelta1), Inhibitor
Full Product Name
Selective PI3Kdelta Inhibitor 1
Product Gene Name
Form/Format
Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.
Molecular Weight
429.45
Formula
C23H20FN7O
CAS
2088525-31-7
Smiles
Cn1nc(nc1C1(CC1)c1ccccc1)-c1cnc(N)c(n1)-c1ccc(C(N)=O)c(F)c1
Receptor (IC50)
PI3Kdelta: 0.9nM
Solubility
DMSO: 43mg/mL (100.13mM)
(<1mg/ml refers to the product slightly soluble or insoluble)

Product References and Citations for PI3Kdelta1, inhibitor

1. Terstiege I, Perry M, Petersen J, et al. Discovery of triazole aminopyrazines as a highly potent and selective series of PI3Kdelta inhibitors[J]. Bioorganic & medicinal chemistry letters, 2016, 27 (3).

Other Notes

Small volumes of PI3Kdelta1, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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