Ezatiostat Inhibitor

Name: Ezatiostat Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5752202
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752202

Ezatiostat is a liposomal small-molecule glutathione analog inhibitor of glutathione S-transferase (GST) P1-1 with hematopoiesis-stimulating activity. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Ezatiostat, Inhibitor

Full Product Name

Ezatiostat

Product Synonym Names

Ezatiostat TFA (free base); TER199 (free base); TLK199

Form/Format

Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Molecular Weight

529.65

Formula

C29H36F3N3O8S

CAS

168682-53-9

Smiles

CCOC(=O)C(N)CCC(=O)NC(CSCc1ccccc1)C(=O)NC(C(=O)OCC)c1ccccc1

Receptor (IC50)

GSTP

Solubility

DMSO: >50mg/mL (94.4mM)
Ethanol: 20mg/mL (37.76)
Water: Insoluble
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for Ezatiostat, inhibitor

Home; Others

Product References and Citations for Ezatiostat, inhibitor

1. Ruscoe J E, Rosario L A, Wang T, et al. Pharmacologic or Genetic Manipulation of Glutathione S-Transferase P1-1 (GSTpi) Influences Cell Proliferation Pathways[J]. Journal of Pharmacology and Experimental Therapeutics, 2001, 298 (1):339-345.
2. Galili N, Tamayo P, Botvinnik O B, et al. Prediction of response to therapy with ezatiostat in lower risk myelodysplastic syndrome[J]. Journal of Hematology & Oncology, 2012, 5 (1):20.

Other Notes

Small volumes of Ezatiostat, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Ezatiostat purchase

MBS5752202 is an inhibitor targeting Ezatiostat.