Valbenazine Inhibitor

Name: Valbenazine Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5752360
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752360

Valbenazine, a highly selective vesicular monoamine transporter 2 (VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Valbenazine, Inhibitor

Full Product Name

Valbenazine

Product Synonym Names

NBI-98854

Form/Format

Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Molecular Weight

418.57

Formula

C24H38N2O4

CAS

1025504-45-3

Smiles

[H][C@]12C[C@@H](OC(=O)[C@@H](N)C(C)C)[C@H](CC(C)C)CN1CCc1cc(OC)c(OC)cc21

Receptor (IC50)

VMAT2

Solubility

DMSO: 50mg/mL (119.45mM)
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for Valbenazine, inhibitor

Home; Membrane transporter/Ion Channel

Product References and Citations for Valbenazine, inhibitor

1. Josiassen R C, Kane J M, Liang G S, et al. Long-Term Safety and Tolerability of Valbenazine (NBI-98854) in Subjects with Tardive Dyskinesia and a Diagnosis of Schizophrenia or Mood Disorder[J]. Psychopharmacology bulletin, 2017, 47 (3):61-68.
2. Factor S A, Remington G, Comella C L, et al. The Effects of Valbenazine in Participants with Tardive Dyskinesia: Results of the 1-Year KINECT 3 Extension Study[J]. The Journal of Clinical Psychiatry, 2017, 78 (9).
3. Müller T, et al. Valbenazine granted breakthrough drug status for treating tardive dyskinesia. Expert Opin Investig Drugs. 2015 Jun;24 (6):737-42.

Other Notes

Small volumes of Valbenazine, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Valbenazine purchase

MBS5752360 is an inhibitor targeting Valbenazine.