AMG9810 Inhibitor

Name: AMG9810 Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5752395
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752395

AMG 9810 is a competitive antagonist of capsaicin activation of the vanilloid receptor 1 (TRPV1) (IC50s = 24.5 and 85.6nM for human and rat TRPV1, respectively). More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

AMG9810, Inhibitor

Full Product Name

AMG9810

Product Gene Name

AMG9810, inhibitor

Form/Format

Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Molecular Weight

337.41

Formula

C21H23NO3

CAS

545395-94-6

Smiles

CC(C)(C)c1ccc(cc1)\C=C\C(=O)Nc1ccc2OCCOc2c1

Receptor (IC50)

hTRPV1: 24.5nM
mTRPV1: 85.6nM

Solubility

DMSO: 33mg/mL (97.80mM)
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for AMG9810, inhibitor

Home; Membrane transporter/Ion Channel

Product References and Citations for AMG9810, inhibitor

1. Mcdougle D R, Watson J E, Abdeen A A, et al. Anti-inflammatory omega-3 endocannabinoid epoxides[J]. Proceedings of the National Academy of Sciences, 2017:201610325.
2. Wolf F I, Vsimonacci T. Effect of transient receptor potential vanilloid 1 (TRPV1) receptor antagonist compounds SB705498, BCTC and AMG9810 in rat models of thermal hyperalgesia measured with an increasing-temperature water bath.[J]. European Journal of Pharmacology, 2010, 641 (2):135-141.

Other Notes

Small volumes of AMG9810, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for AMG9810 purchase

MBS5752395 is an inhibitor targeting AMG9810.