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Mirogabalin Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752419

MBS5752419 is an inhibitor targeting Mirogabalin. Mirogabalin is a calcium channel blocker with analgesic effects. More details

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Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Mirogabalin, Inhibitor
Full Product Name
Mirogabalin
Product Synonym Names
DS5565
Form/Format
Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.
Molecular Weight
209.28
Formula
C12H19NO2
CAS
1138245-13-2
Smiles
[H][C@@]12C[C@](CN)(CC(O)=O)[C@]1([H])C=C(CC)C2
Receptor (IC50)
alpha2delta calcium channels
Solubility
H2O: 7.71mg/mL (36.84mM)
Methanol: 16mg/mL (76.45mM)
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for Mirogabalin, inhibitor

Home; Membrane transporter/Ion Channel

Structure of Mirogabalin, inhibitor

Mirogabalin Inhibitor – Cat# MBS5752419

Product References and Citations for Mirogabalin, inhibitor

1. Vinik A, Rosenstock J, Sharma U, et al. Efficacy and Safety of Mirogabalin (DS-5565) for the Treatment of Diabetic Peripheral Neuropathic Pain: A Randomized, Double-Blind, Placebo- and Active Comparator-Controlled, Adaptive Proof-of-Concept Phase 2 Study[J]. Diabetes Care, 2014, 37 (12):3253-61.
2. HutmachermM, et al. Exposure-response modeling of average daily pain score, and dizziness and somnolence, forMirogabalin (DS-5565) in patients with diabetic peripheral neuropathic pain. J Clin Pharmacol. 2016 Jan;56 (1):67-77.

Other Notes

Small volumes of Mirogabalin, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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