F-15599 Inhibitor

Name: F-15599 Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5752437
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752437

F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist (Ki : 3.4nM). More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

F-15599, Inhibitor

Full Product Name

F-15599

Product Gene Name

F-15599, inhibitor

Form/Format

Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Molecular Weight

394.85

Formula

C19H21ClF2N4O

CAS

635323-95-4

Smiles

Cc1cnc(CNCC2(F)CCN(CC2)C(=O)c2ccc(F)c(Cl)c2)nc1

Receptor (IC50)

5-HT1A: 3.4nM (ki)

Solubility

DMSO: 250mg/mL (633.15mM), Need ultrasonic:
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for F-15599, inhibitor

Home; GPCR/G Protein; 5-HT Receptor

Product References and Citations for F-15599, inhibitor

1. De Boer S F, Newman-Tancredi A. Anti-aggressive effects of the selective high-efficacy 'biased' 5-HT1Areceptor agonists F15599 and F13714 in male WTG rats[J]. Psychopharmacology, 2016, 233 (6):937-947.
2. Preferential in vivo action of F15599, a novel 5-HT1A receptor agonist, at postsynaptic 5-HT1A receptors[J]. British Journal of Pharmacology, 2010, 160 (8):1929-1940.

Other Notes

Small volumes of F-15599, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for F-15599 purchase

MBS5752437 is an inhibitor targeting F-15599.