Ralfinamide Inhibitor

Name: Ralfinamide Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5752492
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752492

Ralfinamide is an orally available Na-channel blocker for the treatment of neuropathic pain and other pain conditions. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Ralfinamide, Inhibitor

Full Product Name

Ralfinamide

Product Synonym Names

FCE-26742A; Priralfinamide

Form/Format

Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Molecular Weight

302.34

Formula

C17H19FN2O2

CAS

133865-88-0

Smiles

C[C@H](NCc1ccc(OCc2ccccc2F)cc1)C(N)=O

Receptor (IC50)

Na-channel

Solubility

DMSO: 125mg/mL (413.44mM)
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for Ralfinamide, inhibitor

Home; Membrane transporter/Ion Channel

Product References and Citations for Ralfinamide, inhibitor

1. Liang X, Yu G, Su R. Effects of ralfinamide in models of nerve injury and chemotherapy-induced neuropathic pain[J]. European journal of pharmacology, 2018, 823:27-34.
2. Zhang S H, Blech-Hermoni Y, Faravelli L, et al. Ralfinamide administered orally before hindpaw neurectomy or postoperatively provided long-lasting suppression of spontaneous neuropathic pain-related behavior in the rat[J]. Pain, 2008, 139 (2):0-305.

Other Notes

Small volumes of Ralfinamide, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Ralfinamide purchase

MBS5752492 is an inhibitor targeting Ralfinamide.