BRD9539 Inhibitor

Name: BRD9539 Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5752513
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752513

BRD9539 is an inhibitor of euchromatin histone methyltransferase 2 (EHMT2), also known as G9a, with an IC50 value of 6.3uM More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

BRD9539, Inhibitor

Full Product Name

BRD9539

Form/Format

Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Molecular Weight

399.44

Formula

C24H21N3O3

CAS

1374601-41-8

Smiles

OC(=O)c1ccc2n(CCCc3ccccc3)c(NC(=O)c3ccccc3)nc2c1

Receptor (IC50)

G9a

Solubility

DMSO: 35mg/mL (87.62mM)
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for BRD9539, inhibitor

Home; Chromatin/Epigenetic; Histone Methyltransferase

Product References and Citations for BRD9539, inhibitor

1. Yuan Y, Wang Q, Paulk J, et al. A Small-Molecule Probe of the Histone Methyltransferase G9a Induces Cellular Senescence in Pancreatic Adenocarcinoma[J]. ACS Chemical Biology, 2012, 7 (7):1152-1157.

Other Notes

Small volumes of BRD9539, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for BRD9539 purchase

MBS5752513 is an inhibitor targeting BRD9539.