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AKR1C3-IN-1 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752530

MBS5752530 is an inhibitor targeting AKR1C3-IN-1. AKR1C3-IN-1 is a potent and selective inhibitor of AKR1C3 (IC50 of 13nM). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
AKR1C3-IN-1, Inhibitor
Full Product Name
AKR1C3-IN-1
Product Gene Name
AKR1C3-IN-1, inhibitor
Form/Format
Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.
Molecular Weight
317.36
Formula
C16H15NO4S
CAS
327092-81-9
Smiles
OC(=O)c1cccc(c1)S(=O)(=O)N1CCc2ccccc2C1
Receptor (IC50)
AKR1C3: 13nM
Solubility
DMSO: 100mg/mL (315.10mM)
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for AKR1C3-IN-1, inhibitor

Home; Metabolism; NADPH

Structure of AKR1C3-IN-1, inhibitor

AKR1C3-IN-1 Inhibitor – Cat# MBS5752530

Product References and Citations for AKR1C3-IN-1, inhibitor

1. Jamieson S M F, Brooke D G, Heinrich D, et al. 3- (3,4-Dihydroisoquinolin-2 (1 H)-ylsulfonyl)benzoic Acids: Highly Potent and Selective Inhibitors of the Type 5 17-beta-Hydroxysteroid Dehydrogenase AKR1C3[J]. Journal of Medicinal Chemistry, 2012, 55 (17):7746-7758.

Other Notes

Small volumes of AKR1C3-IN-1, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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