Melperone Inhibitor

Name: Melperone Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5752536
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752536

Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro. More details

Please Inquire

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Melperone, Inhibitor

Full Product Name

Melperone

Form/Format

Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.

Molecular Weight

263.35

Formula

C16H22FNO

CAS

3575-80-2

Smiles

CC1CCN(CCCC(=O)c2ccc(F)cc2)CC1

Solubility

DMSO: 41.67mg/mL (158.23mM)
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for Melperone, inhibitor

Home; Others

Product References and Citations for Melperone, inhibitor

1. Millar J S, Vaughan Williams E M. Differential actions on rabbit nodal, atrial, Purkinje cell and ventricular potentials of melperone, a bradycardic agent delaying repolarization: effects of hypoxia.[J]. British Journal of Pharmacology, 2012, 75 (1):109-121.
2. Whiskey E, Vavrova M, Gaughran F, et al. Melperone in treatment-refractory schizophrenia: a case series[J]. Therapeutic Advances in Psychopharmacology, 2011, 1 (1):19-23.
3. Hefner G, et al. Melperone but not bisoprolol or metoprolol is a clinically relevant inhibitor of CYP2D6: evidence from a therapeutic drug monitoring survey. J Neural Transm (Vienna). 2015 Nov;122 (11):1609-17.

Other Notes

Small volumes of Melperone, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Melperone purchase

MBS5752536 is an inhibitor targeting Melperone.