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BPR1M97 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752820

BPR1M97 is a dual-acting mu-opioid receptor (MOP) and nociceptin-orphanin FQ peptide (NOP) receptor agonist (Kis: 1.8 and 4.2nM) with blood-brain barrier penetration. It produces potent antinociceptive effects. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
BPR1M97, Inhibitor
Full Product Name
BPR1M97
Product Gene Name
BPR1M97, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
349.25
Solubility
DMSO: 250mg/mL (715.82mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C18H18Cl2N2O
SMILES
O=C(NCC1N(C)CCC2=C1C=CC=C2)C3=CC=C(Cl)C(Cl)=C3
CAS Number
2059904-66-2
Target & IC50
MOP: ic50 1.8nM (ki)
NOP: ic50 4.2nM
In Vitro
In a murine model of cancer pain, BPR1M97 (1.8mg/kg; s.c.; once) demonstrates antinociception.

Product References and Citations for BPR1M97, inhibitor

Chao PK, et al. BPR1M97, a dual mu opioid receptor/nociceptin-orphanin FQ peptide receptor agonist, producespotent antinociceptive effects with safer properties than morphine. Neuropharmacology. 2019 Jul 3:107678.
Chao PK, et al. BPR1M97, a dual mu opioid receptor/nociceptin-orphanin FQ peptide receptor agonist, producespotent antinociceptive effects with safer properties than morphine. Neuropharmacology. 2019 Jul 3:107678.

Other Notes

Small volumes of BPR1M97, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for BPR1M97 purchase

MBS5752820 is an inhibitor targeting BPR1M97.
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