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CAV2.2 Inhibitor – Cav 2.2 Blocker 1

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752867

Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1nM) blocker for the treatment,of pain. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Cav 2.2 blocker 1 (Cav2.2), Inhibitor
Full Product Name
Cav 2.2 blocker 1
Product Gene Name
Cav2.2, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
424.96
Solubility
DMSO: 20.83mg/mL (49.02mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C25H29ClN2O2
SMILES
COC(C=CC=C1)=C1N2C(C3=CC=C(Cl)C=C3)=CC(C4CC(C)(C)OC(C)(C)C4)=N2
CAS Number
1567335-29-8
Target & IC50
Cav 2.2: ic50 1nM

Structure of Cav2.2, inhibitor

CAV2.2 Inhibitor – Cat# MBS5752867

Product References and Citations for Cav2.2, inhibitor

Wall MJ, et al. Discovery and optimization of a novel series of pyrazolyltetrahydropyran N-type calcium channel (Cav 2.2) blockers for the treatment,of pain. Bioorg Med Chem Lett. 2018 Dec 15;28(23-24):3780-3783.
Wall MJ, et al. Discovery and optimization of a novel series of pyrazolyltetrahydropyran N-type calcium channel (Cav 2.2) blockers for the treatment,of pain. Bioorg Med Chem Lett. 2018 Dec 15;28(23-24):3780-3783.

Other Notes

Small volumes of Cav2.2, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Cav2.2 purchase

MBS5752867 is an inhibitor targeting Cav2.2. Also known as Cav 2.2 blocker 1.
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