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CDK8-IN-1 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752890

MBS5752890 is an inhibitor targeting CDK8-IN-1. CDK8-IN-1 is a selective CDK8 inhibitor (IC50: 3nM). More details

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Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
CDK8-IN-1, Inhibitor
Full Product Name
CDK8-IN-1
Product Gene Name
CDK8-IN-1, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
255.2
Solubility
<1mg/ml refers to the product slightly soluble or insoluble
Formula
C11H8F3N3O
SMILES
NC(C1=C(C(F)(F)F)C(C2=CC=NC=C2)=CN1)=O
CAS Number
1629633-48-2
Target & IC50
CDK8: ic50 3nM

Product Categories/Family for CDK8-IN-1, inhibitor

Cell Cycle/Checkpoint; CDK

Structure of CDK8-IN-1, inhibitor

CDK8-IN-1 Inhibitor – Cat# MBS5752890

Product References and Citations for CDK8-IN-1, inhibitor

Han X, et al. Discovery of potent and selective CDK8 inhibitors through FBDD approach. Bioorg Med Chem Lett. 2017 Sep 15;27(18):4488-4492.
Han X, et al. Discovery of potent and selective CDK8 inhibitors through FBDD approach. Bioorg Med Chem Lett. 2017 Sep 15;27(18):4488-4492.

Other Notes

Small volumes of CDK8-IN-1, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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