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CDK9-IN-8 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752895

MBS5752895 is an inhibitor targeting CDK9-IN-8. CDK9-IN-8 is a highly potent and selective CDK9 inhibitor (IC50: 12nM). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
CDK9-IN-8, Inhibitor
Full Product Name
CDK9-IN-8
Product Gene Name
CDK9-IN-8, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
569.63
Solubility
DMSO: 5.2mg/mL (9.13mM) ultrasonic and warming and heat to 80 degree C
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C31H32FN7O3
SMILES
FC1=CC=C(NC(C2(CC2)C(NC3=CC=C(NC4=NC=C5C(N(C6CCCC6)C(C(N(C)C)=O)=C5)=N4)C=C3)=O)=O)C=C1
CAS Number
2105956-51-0
Target & IC50
CDK9: ic50 12nM

Product Categories/Family for CDK9-IN-8, inhibitor

Cell Cycle/Checkpoint; CDK

Structure of CDK9-IN-8, inhibitor

CDK9-IN-8 Inhibitor – Cat# MBS5752895

Product References and Citations for CDK9-IN-8, inhibitor

Li Y, et al. Discovery of a highly potent, selective and novel CDK9 inhibitor as an anticancer drug candidate. Bioorg Med Chem Lett. 2017 Aug 1;27(15):3231-3237.
Li Y, et al. Discovery of a highly potent, selective and novel CDK9 inhibitor as an anticancer drug candidate. Bioorg Med Chem Lett. 2017 Aug 1;27(15):3231-3237.

Other Notes

Small volumes of CDK9-IN-8, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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