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CGP25454A Inhibitor – CGP 25454a

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752911

CGP 25454A is a novel and selective antagonist of the presynaptic dopamine autoreceptor. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
CGP 25454A (CGP25454A), Inhibitor
Full Product Name
CGP 25454A
Product Gene Name
CGP25454A, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
346.25
Solubility
DMSO: 3.5mg/mL (10.11mM)
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C15H21Cl2N3O2
SMILES
O=C(NCCN(CC)CC)C1=CC(C#N)=C(Cl)C=C1OC.[H]Cl
CAS Number
104391-26-6
Target & IC50
Others
In Vitro
CGP 25454A increase [3H]spiperone binding to receptors of the D2 family in rat striatum by 90-110% (ED50: 13mg/kg i.p.). At 30-100mg/kg, CGP 25454A inhibits [3H]spiperone binding in the pituitary of the same animals as a result of a blockade of postsynaptic DA receptors.

Structure of CGP25454A, inhibitor

CGP25454A Inhibitor – Cat# MBS5752911

Product References and Citations for CGP25454A, inhibitor

Bischoff S et al. CGP 25454A, a novel and selective presynaptic dopamine autoreceptor antagonist. Naunyn Schmiedebergs Arch Pharmacol. 1994 Sep;350(3):230-8.
Bischoff S et al. CGP 25454A, a novel and selective presynaptic dopamine autoreceptor antagonist. Naunyn Schmiedebergs Arch Pharmacol. 1994 Sep;350(3):230-8.

Other Notes

Small volumes of CGP25454A, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for CGP25454A purchase

MBS5752911 is an inhibitor targeting CGP25454A. Also known as CGP 25454A.
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