CY208-243 Inhibitor – Cy 208-243

Name: CY208-243 Inhibitor; Cy 208-243; MyBioSource
Brand: MyBioSource
SKU: MBS5752961
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5752961

CY 208-243 is a selective dopamine D1 receptor agonist with anti-Parkinson disease activity. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

CY 208-243 (CY208-243), Inhibitor

Full Product Name

CY 208-243

Product Gene Name

CY208-243, inhibitor

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

274.36

Solubility

<1mg/ml refers to the product slightly soluble or insoluble

Formula

C19H18N2

SMILES

CN1[C@@](C2)([H])[C@@](C3=CC=CC=C3C1)([H])C4=CC=CC5=C4C2=CN5

CAS Number

100999-26-6

Target & IC50

In Vitro

CY 208-243 (2.5 mg/kg; s.c.) pretreatment,prevents D-1 antagonist SCH 23390 (0.05 mg/kg; s.c.)-Induced DA release and increased metabolism.

Product Categories/Family for CY208-243, inhibitor

GPCR/G Protein; Dopamine Receptor; Neuroscience

Product References and Citations for CY208-243, inhibitor

Imperato A, et al. CY 208-243, a novel dopamine D-1 receptor agonist, fails to modify dopamine release in freely moving rats. Eur J Pharmacol. 1989 Jan 24;160(1):155-8.
Temlett JA, et al. The D-1 dopamine receptor partial agonist, CY 208-243, exhibits antiparkinsonian activity in the MPTP-treated marmoset. Eur J Pharmacol. 1988 Nov 1;156(2):197-206.
Temlett JA, et al. The D-1 dopamine receptor partial agonist, CY 208-243, exhibits antiparkinsonian activity in the MPTP-treated marmoset. Eur J Pharmacol. 1988 Nov 1;156(2):197-206.

Other Notes

Small volumes of CY208-243, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for CY208-243 purchase

MBS5752961 is an inhibitor targeting CY208-243. Also known as CY 208-243.