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(R)-Elagolix Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5753081

Elagolix is a selective, highly potent, short-duration, orally-active, non-peptidethe gonadotropin-releasing hormone receptor (GnRHR) antagonist with KD of 54 pM More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
(R)-Elagolix, Inhibitor
Full Product Name
(R)-Elagolix
Product Synonym Names
NBI-56418
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
631.59
Solubility
DMSO: 100mg/mL (158.33mM)
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C32H30F5N3O5
SMILES
FC1=C(C2=C(C)N(CC3=C(C(F)(F)F)C=CC=C3F)C(N(C[C@](C4=CC=CC=C4)([H])NCCCC(O)=O)C2=O)=O)C=CC=C1OC
CAS Number
834153-87-6
Target & IC50
Others

Structure of (R)-Elagolix, inhibitor

(R)-Elagolix Inhibitor – Cat# MBS5753081

Product References and Citations for (R)-Elagolix, inhibitor

Carr B, et al. Elagolix, an oral GnRH antagonist, versus subcutaneous depot medroxyprogesterone acetate for the treatment,of endometriosis: effects on bone mineral density. Reprod Sci. 2014 Nov;21(11):1341-1351.
Carr B, et al. Elagolix, an oral GnRH antagonist, versus subcutaneous depot medroxyprogesterone acetate for the treatment,of endometriosis: effects on bone mineral density. Reprod Sci. 2014 Nov;21(11):1341-1351.

Other Notes

Small volumes of (R)-Elagolix, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for (R)-Elagolix purchase

MBS5753081 is an inhibitor targeting (R)-Elagolix.
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