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Molibresib besylate Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5753232

MBS5753232 is an inhibitor targeting Molibresib besylate. Molibresib besylate is an inhibitor of BET bromodomain (IC50: 32.5-42.5nM). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Molibresib besylate, Inhibitor
Full Product Name
Molibresib besylate
Product Synonym Names
GSK 525762C; I-BET 762 besylate
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
582.07
Solubility
DMSO: 25mg/mL (42.95mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C28H28ClN5O5S
SMILES
ClC1=CC=C(C2=N[C@@H](CC(NCC)=O)C3=NN=C(C)N3C4=CC=C(OC)C=C24)C=C1.O=S(C5=CC=CC=C5)(O)=O
CAS Number
1895049-20-3
Target & IC50
BET: ic50 32.5-42.5nM

Product Categories/Family for Molibresib besylate, inhibitor

Immunology/Inflammation; CCR; Chromatin/Epigenetic; Epigenetics

Structure of Molibresib besylate, inhibitor

Molibresib besylate Inhibitor – Cat# MBS5753232

Product References and Citations for Molibresib besylate, inhibitor

Nicodeme E, et al. Suppression of inflammation by a synthetic histone mimic. Nature. 2010 Dec 23;468(7327):1119-23.

Other Notes

Small volumes of Molibresib besylate, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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