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GV-58 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5753262

GV-58 is a selective N- and P/Q-type Ca2+ channels agonist (EC50: 7.21/8.81uM for N-type/P-Q-type Ca2+ channel). The inhibitory of GV-58 is 20-fold fewer for CDK kinases activity. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
GV-58, Inhibitor
Full Product Name
GV-58
Product Gene Name
GV-58, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
374.5
Solubility
DMSO: 50mg/mL (133.51mM) Need ultrasonic
H2O: <0.1mg/mL (insoluble)
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C18H26N6OS
SMILES
CC[C@@H](NC1=NC(NCC2=CC=C(C)S2)=C3N=CN(CCC)C3=N1)CO
CAS Number
1402821-41-3
Target & IC50
Others

Structure of GV-58, inhibitor

GV-58 Inhibitor – Cat# MBS5753262

Product References and Citations for GV-58, inhibitor

Tarr TB, et al. Evaluation of a novel calcium channel agonist for therapeutic potential in Lambert-Eaton myasthenic syndrome. J Neurosci. 2013 Jun 19;33(25):10559-67.
Tarr TB, et al. Evaluation of a novel calcium channel agonist for therapeutic potential in Lambert-Eaton myasthenic syndrome. J Neurosci. 2013 Jun 19;33(25):10559-67.

Other Notes

Small volumes of GV-58, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GV-58 purchase

MBS5753262 is an inhibitor targeting GV-58.
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