KHK-IN-2 Inhibitor

Name: KHK-IN-2 Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5753366
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5753366

KHK-IN-2 is a selective and potent ketohexokinase (KHK) inhibitor with an IC50 of 0.45uM. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

KHK-IN-2, Inhibitor

Full Product Name

KHK-IN-2

Product Gene Name

KHK-IN-2, inhibitor

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

372.34

Solubility

DMSO: 250mg/mL (671.43mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)

Formula

C16H19F3N4O3

SMILES

N#CC1=C(C(F)(F)F)C=C(N2C[C@H](O)[C@@H](O)C2)N=C1N3CC[C@](C)(O)C3

CAS Number

2135304-43-5

Target & IC50

KHK: ic50 0.45uM

Product Categories/Family for KHK-IN-2, inhibitor

Chromatin/Epigenetic; Histone Demethylase; Others

Product References and Citations for KHK-IN-2, inhibitor

Huard K, et al. Discovery of Fragment-Derived Small Molecules for in Vivo Inhibition of Ketohexokinase (KHK). J Med Chem. 2017 Sep 28;60(18):7835-7849.

Other Notes

Small volumes of KHK-IN-2, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for KHK-IN-2 purchase

MBS5753366 is an inhibitor targeting KHK-IN-2.