LAU159 Inhibitor

Name: LAU159 Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5753392
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5753392

LAU159 is a functionally selective positive alpha1beta3 GABA(A) receptor modulator(EC50 : 2.2uM). More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

LAU159, Inhibitor

Full Product Name

LAU159

Product Gene Name

LAU159, inhibitor

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

325.75

Solubility

<1mg/ml refers to the product slightly soluble or insoluble

Formula

C17H12ClN3O2

SMILES

COc1cccc(c1)-n1[nH]c2c(cnc3ccc(Cl)cc23)c1=O

CAS Number

2055050-87-6

Target & IC50

alpha1beta3 GABA: ic50 2.2uM (EC50)

Product Categories/Family for LAU159, inhibitor

Membrane transporter/Ion channel; Neuroscience

Product References and Citations for LAU159, inhibitor

Varagic Z, et al. Identification of novel positive allosteric modulators and null modulators at the GABAA receptor alpha+beta- interface. Br J Pharmacol. 2013 May;169(2):371-83.

Other Notes

Small volumes of LAU159, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for LAU159 purchase

MBS5753392 is an inhibitor targeting LAU159.