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OXFBD04 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5753630

MBS5753630 is an inhibitor targeting OXFBD04. OXFBD04 is a potent and selective inhibitor of BRD4(IC50 of 166nM). More details

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Product Documentation
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Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
OXFBD04, Inhibitor
Full Product Name
OXFBD04
Product Gene Name
OXFBD04, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
296.32
Solubility
DMSO: 250mg/mL (843.68mM)
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C17H16N2O3
SMILES
OC(C1=CC(O)=CC(C2=C(C)ON=C2C)=C1)C3=CC=CN=C3
CAS Number
2231747-03-6
Target & IC50
BRD4: ic50 166nM

Product Categories/Family for OXFBD04, inhibitor

Chromatin/Epigenetic; Epigenetic Reader Domain

Structure of OXFBD04, inhibitor

OXFBD04 Inhibitor – Cat# MBS5753630

Product References and Citations for OXFBD04, inhibitor

Jennings LE, et al. BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability. Bioorg Med Chem. 2018 Jul 15;26(11):2937-2957.
Jennings LE, et al. BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability. Bioorg Med Chem. 2018 Jul 15;26(11):2937-2957.

Other Notes

Small volumes of OXFBD04, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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