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Pentiapine Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5753660

MBS5753660 is an inhibitor targeting Pentiapine. Pentiapine is a novel inhibitor of dopamine release. More details

Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Pentiapine, Inhibitor
Full Product Name
Pentiapine
Product Synonym Names
CGS 10746
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
299.39
Solubility
DMSO: 100mg/mL (334.01mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C15H17N5S
SMILES
CN1CCN(C2=NC3=CC=CC=C3SC4=NC=CN42)CC1
CAS Number
81382-51-6
Target & IC50
Dopamine
In Vitro
Pentiapine dose-dependently reduces motor activity of mice.

Product References and Citations for Pentiapine, inhibitor

Manzanedo C, et al. Effects of CGS 10746B on hyperactivity and place preference induced by morphine. Behav Brain Res. 2001 Nov 29;126(1-2):23-32.
Manzanedo C, et al. Effects of CGS 10746B on hyperactivity and place preference induced by morphine. Behav Brain Res. 2001 Nov 29;126(1-2):23-32.
Bilsky EJ, et al. CGS 10746B, a novel dopamine release inhibitor, blocks the establishment of cocaine and MDMA conditioned place preferences. Pharmacol Biochem Behav. 1998 Jan;59(1):215-20.
Bilsky EJ, et al. CGS 10746B, a novel dopamine release inhibitor, blocks the establishment of cocaine and MDMA conditioned place preferences. Pharmacol Biochem Behav. 1998 Jan;59(1):215-20.

Other Notes

Small volumes of Pentiapine, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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