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PX20606 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5753747

PX20606 trans racemate is an agonist of FXR (EC50s of 32 and 34nM for FXR in FRET and M1H assay, respectively). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
PX20606, Inhibitor
Full Product Name
PX20606 trans racemate
Product Gene Name
PX20606, inhibitor
Product Synonym Names
PX-102 trans racemate
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
554.85
Solubility
<1mg/ml refers to the product slightly soluble or insoluble
Formula
C29H22Cl3NO4
SMILES
O=C(O)C1=CC=C([C@H]2[C@H](C3=CC=C(OCC4=C(C5CC5)ON=C4C6=C(Cl)C=CC=C6Cl)C=C3Cl)C2)C=C1.[relative sterochemistry]
CAS Number
1268244-85-4
Target & IC50
Others

Product References and Citations for PX20606, inhibitor

Kinzel O, et al. Novel substituted isoxazole FXR agonists with cyclopropyl, hydroxycyclobutyl and hydroxyazetidinyl linkers: Understanding and improving key determinants of pharmacological properties. Bioorg Med Chem Lett. 2016 Aug 1;26(15):3746-53.
Kinzel O, et al. Novel substituted isoxazole FXR agonists with cyclopropyl, hydroxycyclobutyl and hydroxyazetidinyl linkers: Understanding and improving key determinants of pharmacological properties. Bioorg Med Chem Lett. 2016 Aug 1;26(15):3746-53.

Other Notes

Small volumes of PX20606, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for PX20606 purchase

MBS5753747 is an inhibitor targeting PX20606. Also known as PX20606 trans racemate.
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