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(R)-BAY-85-8501 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5753763

(R)-BAY-85-8501 is the less active enantiomer of BAY-85-8501. BAY-85-8501 is a selective and potent Human Neutrophil Elastase (HNE)inhibitor(IC50 of 65 pM). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
(R)-BAY-85-8501, Inhibitor
Full Product Name
(R)-BAY-85-8501
Product Gene Name
(R)-BAY-85-8501, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
474.46
Solubility
<1mg/ml refers to the product slightly soluble or insoluble
Formula
C22H17F3N4O3S
SMILES
N#CC1=C(C)N(C2=CC=CC(C(F)(F)F)=C2)C(N(C)[C@H]1C3=CC=C(C#N)C=C3S(=O)(C)=O)=O
Target & IC50
Others

Structure of (R)-BAY-85-8501, inhibitor

(R)-BAY-85-8501 Inhibitor – Cat# MBS5753763

Product References and Citations for (R)-BAY-85-8501, inhibitor

Von Nussbaum F, et al. Freezing the Bioactive Conformation to Boost Potency: The Identification of BAY 85-8501, a Selective and Potent Inhibitor of Human Neutrophil Elastase for Pulmonary Diseases. ChemMedChem. 2015 Jul;10(7):1163-73.
Von Nussbaum F, et al. Freezing the Bioactive Conformation to Boost Potency: The Identification of BAY 85-8501, a Selective and Potent Inhibitor of Human Neutrophil Elastase for Pulmonary Diseases. ChemMedChem. 2015 Jul;10(7):1163-73.

Other Notes

Small volumes of (R)-BAY-85-8501, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for (R)-BAY-85-8501 purchase

MBS5753763 is an inhibitor targeting (R)-BAY-85-8501.
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