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RR-11a Inhibitor – Analog

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5753835

RR-11a analog is a potent and selective asparaginyl endopeptidases (AE) (Legumain) inhibitors(IC50 values of 4.5nM, 4.5nM and 31nM for AE1 in Trichomonas Vaginalis, AE in Ixodes ricinus and AE in Schistosoma mansoni, respectively). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
RR-11a analog, Inhibitor
Full Product Name
RR-11a analog
Product Gene Name
RR-11a, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
491.49
Solubility
DMSO: 125mg/mL (254.33mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C22H29N5O8
SMILES
O=C(N[C@@H](C)C(N[C@@H](C)C(NN(CC(N)=O)C(/C=C/C(OCC)=O)=O)=O)=O)OCC1=CC=CC=C1
CAS Number
685543-66-2
Target & IC50
AE1 in Trichomonas Vaginalis: ic50 4.5nM
AE in Ixodes ricinus: ic50 4.5nM
AE in Schistosoma mansoni: ic50 31nM

Structure of RR-11a, inhibitor

RR-11a Inhibitor – Cat# MBS5753835

Product References and Citations for RR-11a, inhibitor

Gotz MG, et al. Aza-peptidyl Michael acceptors. A new class of potent and selective inhibitors of asparaginyl endopeptidases (legumains) from evolutionarily diverse pathogens. J Med Chem. 2008 May 8;51(9):2816-32.

Other Notes

Small volumes of RR-11a, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for RR-11a purchase

MBS5753835 is an inhibitor targeting RR-11a. Also known as RR-11a analog.
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