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SGC-iMLLT Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5753898

SGC-iMLLT is a potent and selective MLLT1/3-histone interactions inhibitor(IC50 of 0.26uM), and is a first-in-class chemical probe. More details

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Product Documentation
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Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
SGC-iMLLT, Inhibitor
Full Product Name
SGC-iMLLT
Product Gene Name
SGC-iMLLT, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
388.47
Solubility
DMSO: 83.33mg/mL (214.51mM) Need ultrasonic
H2O: <0.1mg/mL (insoluble)
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C22H24N6O
SMILES
CN1N=CC2=CC(C(NC3=CC=C(NC(CN4[C@@H](C)CCC4)=N5)C5=C3)=O)=CC=C21
CAS Number
2255338-25-9
Target & IC50
MLLT1 YD: ic50 0.129?uM
MLLT3 YD: ic50 0.077?uM (kd)

Structure of SGC-iMLLT, inhibitor

SGC-iMLLT Inhibitor – Cat# MBS5753898

Product References and Citations for SGC-iMLLT, inhibitor

Moustakim M, et al. Discovery of an MLLT1/3 YEATS Domain Chemical Probe. Angew Chem Int Ed Engl. 2018 Dec 10;57(50):16302-16307.

Other Notes

Small volumes of SGC-iMLLT, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for SGC-iMLLT purchase

MBS5753898 is an inhibitor targeting SGC-iMLLT.
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